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SCI-SSCI veya SCI Expanded Kapsamındaki Yayınları

  • YILMAZ, S., ALTINKANAT-GELMEZ, G., BOLELLI, K., GUNESER-MERDAN, D., OVER-HASDEMIR, M.U., AKI-YALCIN, E., YALCIN, I. "Binding Site Feature Description of 2-Substituted Benzothiazoles as AcrAB-TolC Efflux Pump Inhibitors in E. coli", SAR and QSAR in Environmental Research, 26(10), 853-871
  • ATAEI, S., YILMAZ, S., ERTAN-BOLELLI, T., YILDIZ, I., "Generated 3D-Common Feature Hypotheses Using the HipHop Method For Developing New Topoisomerase I Inhibitors", Archiv der Pharmazie, 348(7), 498-507
  • ZILIFDAR, F., ALPER-HAYTA, S., YILMAZ, S., KAPLAN-OZEN, C., FOTO, E., AYDOGAN, Z., YILDIZ, I., AKI, E., YALCIN, I., DIRIL, N., "Genotoxic potentials and eukaryotic DNA topoisomerase I inhibitory effects of some benzoxazine derivatives", Med. Chem. Res., 23(1), 480-486
  • YILMAZ, S., ALTINKANAT-GELMEZ, G., BOLELLI, K., GUNESER-MERDAN, D., OVER-HASDEMIR, M. U., YILDIZ, I., AKI-YALCIN, E., YALCIN, I., “Pharmacophore Generation of 2-Substituted Benzothiazoles as AdeABC Efflux Pump Inhibitors in A. baumannii”, SAR and QSAR in Environmental Research, 25(7), 551-563
  • ERTAN-BOLELLI, T., MUSDAL, Y., BOLELLI, K., YILMAZ, S., AKSOY, Y., YILDIZ, I., AKI-YALCIN, E., YALCIN, I., “Synthesis, Biological Evaluation of 2-Substituted-5-(4-nitrophenylsulfonamido) benzoxazoles as Human GST P1-1 Inhibitors and Description of the Binding Site Features”, ChemMedChem,9(5), 984-992
  • MUSDAL, Y., ERTAN-BOLELLI, T., BOLELLI, K., YILMAZ, S., CEYHAN, D., HEGAZY, U., MANNERVIK, B., AKSOY, Y., "Inhibition of human glutathione transferase P1-1 by novel benzazole derivatives", Turk. J. Biochem., 37(4), 431-436
  • BHAGYASREE, J.B., VARGHESE, H.T., PANICKER, C.Y., SAMUEL, J., VAN ALSENOY, C., YILMAZ, S., YILDIZ, I., AKI, E., "Quantum mechanical and spectroscopic (FT-IR, FT-Raman, 1H NMR and UV) investigations of 2-(p-nitrobenzyl) benzoxazole", Journal of Molecular Structure, 1046, 92-100
  • YILMAZ, S., YALCIN, I., KAYNAK-ONURDAG, F., OZGEN, S., YILDIZ, I., and AKI, E., "Synthesis and In vitro Antimicrobial Activity of Novel 2-(4-(Substituted-carboxamido)benzyl / phenyl)benzothiazoles", Croat. Chem. Acta, 86(2), 223-231
  • TASKIN, T., YILMAZ, S., YILDIZ, I., YALCIN, I., AKI, E., "Insight into eukaryotic topoisomerase II-inhibiting fused heterocyclic compounds in human cancer cell lines by molecular docking", SAR and QSAR Environmental Research, 23(3-4), 345-355

Uluslararası Bilimsel Toplantılarda Sunulan ve Bildiri Kitabında Basılan Bildiriler (Proceedings)

  • Esin Aki-Yalcin, Serap Yılmaz, Suzan Okten, Fatma Kaynak-Onurdag, Ismail Yalcin. Drug Design Studies of Some Heterocyclic Compounds Active in Hospital-Acquired Infections, 5th International BAU Drug Design Congress, Bahçeşehir University, School of Medicine, Istanbul, Turkey, IS-19: p28, 19-21 October 2017. (Ekim 2017)
  • Ismail Yalcin, Serap Yılmaz, Kayhan Bolelli, Ozum Ozturk, Esin Aki-Yalcin. Structure-Activity Relationship Analysis of Some Benzazoles as Topo II Enzyme Inhibitors, 5th International BAU Drug Design Congress, Bahçeşehir University, School of Medicine, Istanbul, Turkey, IS-18: p27, 19-21 October 2017. (Ekim 2017)
  • Ilkay Yildiz, Sanaz Ataei, Serap Yilmaz, Tugba Ertan-Bolelli, Egemen Foto. Benzoxazine Derivatives as Antitumor Agents Targeting Topo I, 3rd International Turkic World Conference on Chemical Sciences and Technologies (ITWCCST2017), Baku, Azerbaijan, OR-45: p55, September 10-13, 2017. (Eylül 2017)
  • Esin Aki-Yalcin, Serap Yilmaz, Semiha Okten, Fatma Kaynak-Onurdag, Ismail Yalcin. Molecular Docking Studies of 1,4-Benzoxazine Derivatives Against Acinetobacter Baumannii, 11th AFMC International Medicinal Chemistry Symposium (AIMECS2017), Melbourne, Australia, p129, 23-26 July 2017. (Temmuz 2017)
  • Serap Yilmaz, Suzan Okten, Fatma Kaynak-Onurdag, Esin Aki-Yalcin, Ismail Yalcin. Pharmacophore Modeling of 1,4-Benzoxazine Derivatives as Bacterial Topoisomerase II Inhibitors , 17th Hellenic Symposium on Medicinal Chemistry (HSMC-2017), Aristotle University of Thessaloniki, Thessaloniki, Greece, P69: p111, 1-3 June 2017. (Haziran 2017)
  • Ismail Yalcin*, Serap Yilmaz, Kayhan Bolelli, Esin Aki-Yalcin. Binding Site Description Studies of 2-Substituted Benzothiazoles as the Novel RND Efflux Pump Inhibitors, 4rd International Conference on Computation for Science and Technology (ICCST) 2016, De Baron Resort, Langkawi, Malaysia, PLN5: p49, 3-4 November 2016. (Kasım 2016)
  • Egemen Foto, Fatma Zilifdar, Serap Yilmaz, Ismail Yalcin, Nuran Diril. Investigation of Cytotoxic, Genotoxic, Mutagenic Potentials of a Serial 1,4-Benzoxazine-3-one Derivative Compounds and Pharmacophore Modelling, International Conference On Biological Sciences (ICBS), Konya, Turkey, PP-34: p134, October 21-23, 2016. (Ekim 2016)
  • Egemen Foto, Fatma Zilifdar, Serap Yilmaz, Tulay Saracbasi, Ismail Yalcin, Nuran Diril. Mutagenicity of a series efficacious benzoxazine derivatives – a new approach to evaluate ames test data, 41st FEBS Congress, Ephesus, Kusadasi, Aydin, Turkey, P-MIS-080: p186, 03-08 September 2016. (Eylül 2016)
  • Serap Yilmaz, Suzan Okten, Fatma Kaynak Onurdag, Esin Aki Yalcin, Ismail Yalcin. Molecular docking studies of 1,4-benzoxazine derivatives as bacterial topoisomerase II inhibitors, 21st European Symposium on Quantitative Structure-Activity Relationships (21st EuroQSAR), Aptuit Conference Center, Verona, Italy, P008: p89, September 4-8, 2016. (Eylül 2016)
  • Serap Yilmaz, Suzan Okten, Fatma Kaynak Onurdag, Esin Aki Yalcin, Ismail Yalcin. Synthesis and Antibacterial Activity of Some Novel Benzothiazole Derivatıves Holding 1,4-Benzoxazine Ring, 15th Belgian Organic Synthesis Symposium (BOSS XV), Antwerp, Belgium, P011: p66, July 10-15, 2016. (Temmuz 2016)
  • Ismail Yalcin, Serap Yilmaz, Kayhan Bolelli, Esin Aki-Yalcin, Ufuk Over-Hasdemir. Binding site description of 2-substituted benzothiazoles as potential RND efflux pump inhibitors, 6th Congress of Pharmacy in Macedonia, Ohrid, Macedonia, S6 PP 259: p543-544, June 1-5, 2016. (Haziran 2016)
  • Esin Akı Yalçın*, Serap Yılmaz, Kayhan Bolelli, Özüm Öztürk, Tuğba Ertan-Bolelli, İsmail Yalçın, The Role of Chemometrics in Computer Aided Drug Design Studies, 3rd International Conference on New Trends in Chemometrics and Applications (NTCA-2016), Side, Antalya, Turkey, IL-02: p4, May 25-28, 2016. (Mayıs 2016)
  • Egemen Foto, Fatma Zilifdar, Serap Yilmaz, Ismail Yalcin, Nuran Diril. Assessment of Selectivity of A Serial 1,4-Benzoxazine-3-one Derivatives Induced Oxidative DNA Damage on Cancer Cells Using The Modified Alkaline Comet Assay, 2nd International Congress & Workshop of Forensic Toxicology (2nd ForeTox 2016), Ankara, Turkey, P199: p277, May 26-30, 2016. (Mayıs 2016)
  • Kayhan Bolelli, Tugba Ertan-Bolelli, Serap Yilmaz, Ozum Ozturk, Esin Aki-Yalcin, Ismail Yalcin. Pharmacophore Identification Analysis on hGST P1-1 Enzyme Inhibitory Active Benzothiazole Derivatives, Challenges in Organic Chemistry (ISACS19), Irvine, Los Angeles, California, USA, P33, 20-23 March 2016. (Mart 2016)
  • Tugba Ertan-Bolelli, Yaman Musdal, Bengt Mannervik, Kayhan Bolelli, Serap Yilmaz, Ozum Ozturk, Ilkay Yildiz, Esin Aki-Yalcin, Ismail Yalcin. Design and Synthesis of Novel sulfonamide-containing benzoxazoles as Human GST P1-1 Inhibitors, Challenges in Organic Chemistry (ISACS19), Irvine, Los Angeles, California, USA, P15, 20-23 March 2016. (Mart 2016)
  • Serap Yilmaz, Ozum Ozturk, Kayhan Bolelli, Tugba Ertan Bolelli, Esin Aki Yalcin, Ismail Yalcin. Molecular Docking Studies of Some Novel Bacterial Topoisomerase II Inhibitors, The International Chemical Congress of Pacific Basin Societies 2015 (Pacifichem-2015), Honolulu, Hawaii, USA, 10-HLTH-454: p295, 15-20 December 2015. (Aralık 2015)
  • Ozum Ozturk, Esin Aki-Yalcin, Tugba Ertan-Bolelli, Kayhan Bolelli, Serap Yilmaz, Ismail Yalcin. Molecular Modeling Studies of Neurokinin-1 Receptor Antagonists, The International Chemical Congress of Pacific Basin Societies 2015 (Pacifichem-2015), Honolulu, Hawaii, USA, 10-HLTH-450: p294, 15-20 December 2015. (Aralık 2015)
  • Ilkay Yildiz, Tugba Ertan-Bolelli, Sanaz Ataei, Serap Yilmaz, Egemen Foto, Nuran Diril, Ismail Yalcin. Molecular Modeling Studies Topoisomerase I Inhibitors, 3rd International BAU-Drug Design Symposium 2015, Bahçeşehir University, Faculty of Medicine, Istanbul, Turkey, CL-28: p47-48, 1-3 October 2015. (Ekim 2015)
  • Ismail Yalcin, Serap Yilmaz, Gulsen Altinkanat-Gelmez, Kayhan Bolelli, Deniz Guneser-Merdan, M. Ufuk Over-Hasdemir, Esin Aki-Yalcin. Binding Site Description Of Benzothiazoles As the RND Efflux Pump Acrb Inhibitors, 3rd International BAU-Drug Design Symposium 2015, Bahçeşehir University, Faculty of Medicine, Istanbul, Turkey, CL-14: p30, 1-3 October 2015. (Ekim 2015)
  • E. Aki-Yalcin, O. Ozturk, T. Ertan-Bolelli, K. Bolelli, S. Yilmaz, A. H. Nur, O. Bingol-Ozakpinar, and F. Ozdemir. Mechanism of Action of Some New Anticancer Active Neurokinin-1 (NK1) Receptor Antagonists, 10th AFMC International Medicinal Chemistry Symposium (AIMECS 2015), International Convention Center Jeju, Jeju, Korea, OP4-4: p256, 18-21 October 2015. (Ekim 2015)
  • Ismail Yalcin, Serap Yilmaz, Kayhan Bolelli, Ozum Ozturk and Tugba Ertan Bolelli. Enzyme Binding Site Description of AcrAB-TolC Efflux Pump Inhibitors, 10th AFMC International Medicinal Chemistry Symposium (AIMECS 2015), International Convention Center Jeju, Jeju, Korea, OP4-1: p253, 18-21 October 2015. (Ekim 2015)
  • Serap Yilmaz, Ozum Ozturk, Kayhan Bolelli, Tugba Ertan Bolelli, Esin Aki Yalcin, Ismail Yalcin. Pharmacophore Generation of Some Novel Benzothiazole Derivatives as Bacterial Topoisomerase II Inhibitors, 10th AFMC International Medicinal Chemistry Symposium (AIMECS 2015), International Convention Center Jeju, Jeju, Korea, PP2-39: p293, 18-21 October 2015. (Ekim 2015)
  • Esin Akı-Yalcin, Ozum Ozturk, Tugba Ertan-Bolelli, Kayhan Bolelli, Serap Yilmaz, A.H. Nur, S. Sahin, Ismail Yalcin, Ozlem Bingol-Ozakpinar, Filiz Ozdemir. Molecular Modeling Studies on Neurokinin 1 (NK1) Receptors, 8th International Symposium on Computational Methods in Toxicology and Pharmacology Integrating Internet Resources (CMTPI-2015), Chios, Greece, MT-12: p47, 21-25 June 2015. (Haziran 2015)
  • Ilkay Yildiz, Sanaz Ataei, Serap Yilmaz, Tugba Ertan-Bolelli, Egemen Foto, Ismail Yalcin. Pharmacophore Analysis and Molecular Docking Studies on Benzoxazines as Topoisomerase I Inhibitors, 8th International Symposium on Computational Methods in Toxicology and Pharmacology Integrating Internet Resources (CMTPI-2015), Chios, Greece, OC-22: p46, 21-25 June 2015. (Haziran 2015)
  • Ismail Yalcin, Serap Yilmaz, Kayhan Bolelli, Ozum Ozturk, Tugba Ertan-Bolelli, Esin Aki-Yalcin. Description of the Binding Site Features of AcrAB-TolC Efflux Pump Inhibitors, 8th International Symposium on Computational Methods in Toxicology and Pharmacology Integrating Internet Resources (CMTPI-2015), Chios, Greece, MT-11: p44, 21-25 June 2015. (Haziran 2015)
  • E. Foto, F. Zilifdar, S. Yilmaz, N. Diril, I. Yalcin, I. Yildiz, E. Aki Yalcin. Evaluation of In Vitro Genotoxic Potentials of 4-Methyl-6-Substituted-2H-3,4-Dihydro-1,4-Benzoxazin-3-one Derivatives on HeLa Cells, 11th International Symposium on Pharmaceutical Sciences (ISOPS-11), Ankara, Turkey P-382: p427, June 09-12, 2015. (Haziran 2015)
  • E. Foto, F. Zilifdar, N. Diril, S. Yilmaz, E. Aki Yalcin. Mutagenicity of 4-Ethyl-6-substituted-2H-3,4-dihydro-1,4-benzoxazin-3-one Derivatives and Their Metabolites that Inhibited Human Topoisomerase I, 11th International Symposium on Pharmaceutical Sciences (ISOPS-11), Ankara, Turkey P-381: p426, June 09-12, 2015. (Haziran 2015)
  • Sanaz Ataei, Yasin Bayrak, Serap Yilmaz, Tugba Ertan-Bolelli, Ilkay Yildiz. Molecular Studies on Benzazole Derivatives as HIV-1 Reverse Transcriptase Inhibitors, 8th International Symposium on Computational Methods in Toxicology and Pharmacology Integrating Internet Resources (CMTPI-2015), Chios, Greece, PO-2-17: p70, 21-25 June 2015. (Haziran 2015)
  • Serap Yilmaz, Ozum Ozturk, Kayhan Bolelli, Tugba Ertan-Bolelli, Dilara Eren, Esin Aki-Yalcin, Ismail Yalcin. Comparison of Pharmacophore Models between Fluoroquinolones and Nonfluoroquinolone Bacterial Type II Topoisomerase Inhibitors, 8th International Symposium on Computational Methods in Toxicology and Pharmacology Integrating Internet Resources (CMTPI-2015), Chios, Greece, PO-2-14: p67, 21-25 June 2015. (Haziran 2015)
  • Ozum Ozturk, Esin Aki-Yalcin, Tugba Ertan-Bolelli, Kayhan Bolelli, Serap Yilmaz, Ismail Yalcin. Common Pharmacophore Generation of Some Antitumor Agents, 8th International Symposium on Computational Methods in Toxicology and Pharmacology Integrating Internet Resources (CMTPI-2015), Chios, Greece, PO-1-02: p55, 21-25 June 2015. (Haziran 2015)
  • Esin Aki-Yalcin, Ismail Yalcin, Tugba Ertan-Bolelli, Serap Yilmaz, Kayhan Bolelli, Özüm Öztürk, Tugba Taskin-Tok, Emine Öksüzoglu, Cigdem Özen-Kaplan. Computer aided drug design studies for new anticancer drugs, EACR-Sponsored 3rd Anticancer Agent Development Congress, Dokuz Eylül University, Izmir, Turkey, Closing Lecture: p38, 18-19 May 2015. (Mayıs 2015)
  • Ilkay Yildiz, Tugba Ertan-Bolelli, Sanaz Ataei, Serap Yilmaz, Esin Karatas, Kayhan Bolelli, Ozum Ozturk, Ismail Yalcin. Molecular Docking and Pharmacophore Analysis on some Topoisomerase I Targetted Antitumor Benzoxazole and Analogues, 9th Drug Design & Medicinal Chemistry, Berlin, Germany, 5-6 May 2015. (Mayıs 2015)
  • Ozum Ozturk, Esin Akı-Yalçın, Tuğba Ertan-Bolelli, Kayhan Bolelli, Serap Yılmaz, İsmail Yalçın. Pharmacophore generation of neurokinin-1 receptor antagonists as antitumor agents, EACR-Sponsored 3rd Anticancer Agent Development Congress, Dokuz Eylül University, Izmir, Turkey, PP-094: p151, 18-19 May 2015. (Mayıs 2015)
  • Ilkay Yildiz, Sanaz Ataei, Serap Yilmaz, Tugba Ertan-Bolelli, Egemen Foto. Molecular Modeling Studies on BS10 as Topoisomerase I Poison, 1st International Congress: from drug discovery to drug delivery, Royal Olympic Hotel, Athens, Greece, OP-02: p14, 13-15 November 2014. (Kasım 2014)
  • Serap Yilmaz, Tugba Ertan-Bolelli, Kayhan Bolelli, Ozum Ozturk, Sanaz Ataei, Ilkay Yildiz, Esin Aki-Yalcin, Ismail Yalcin. Computational Drug Design Studies for Multidrug Resistance AcrAB-TolC Efflux Pump Inhibitors on Escherichia coli, The 3rd International Conference on Computation for Science and Technology, Aston Denpasar Hotel and Convention Center, Bali, Indonesia, O-P106: p62, 23-25 September 2014. (Eylül 2014)
  • Tugba Ertan-Bolelli, Ismail Yalcin, Yaman Musdal, Serap Yilmaz, Kayhan Bolelli, Ozum Ozturk, Yasemin Aksoy, Bengt Mannervik, Ilkay Yildiz, Esin Aki-Yalcin. Molecular Docking Studies on Human Glutathione S-transferase Enzyme (hGSTP1-1), The 3rd International Conference on Computation for Science and Technology, Aston Denpasar Hotel and Convention Center, Bali, Indonesia, O-P13: p28, 23-25 September 2014. (Eylül 2014)
  • Esin Aki-Yalcin, Tugba Ertan-Bolelli, Kayhan Bolelli, Serap Yilmaz, Ozum Ozturk, Tugba Taskin-Tok, Andry Nur Hidayat, Ilkay Yildiz, Ismail Yalcin. Anticancer Drug Design Studies using Molecular Modeling Techniques, The 3rd International Conference on Computation for Science and Technology, Aston Denpasar Hotel and Convention Center, Bali, Indonesia, IS-02: p10, 23-25 September 2014 (Eylül 2014)
  • Ismail Yalcin, Tugba Ertan-Bolelli, Yaman Musdal, Kayhan Bolelli, Serap Yilmaz, Yasemin Aksoy, Bengt Mannervik, Ilkay Yildiz, Esin Aki-Yalcin. Computer Aided Molecular Modeling of the Binding Site and GSH Conjugation Features of the New Human GST P1-1 Inhibitors, The 3rd International Conference on Computation for Science and Technology, Aston Denpasar Hotel and Convention Center, Bali, Indonesia, PL-03: p6, 23-25 September 2014. (Eylül 2014)
  • Ozum Ozturk, Esin Aki-Yalcin, Tugba Ertan-Bolelli, Kayhan Bolelli, Serap Yilmaz, Ilkay Yildiz, Ismail Yalcin. Common Feature Pharmacophore Generation of Neurokinin-1 Receptor Antagonists, The 3rd International Conference on Computation for Science and Technology, Aston Denpasar Hotel and Convention Center, Bali, Indonesia, P-P110: p103, September 23-25, 2014. (Eylül 2014)
  • Kayhan Bolelli, Ismail Yalcin, Tugba Ertan-Bolelli, Serap Yilmaz, Ozum Ozturk, Ilkay Yildiz, Esin Aki-Yalcin. Pharmacophore Identification Analysis on hGST P1-1 Enzyme Inhibitory Active Benzazole Derivatives, The 3rd International Conference on Computation for Science and Technology, Aston Denpasar Hotel and Convention Center, Bali, Indonesia, P-P12: p76, September 23-25, 2014. (Eylül 2014)
  • Esin Aki-Yalcin, Tugba Ertan-Bolelli, Tugba Taskin-Tok, Cigdem Ozen, Kayhan Bolelli, Serap Yilmaz, Ozum Ozturk, Ilkay Yildiz, Ismail Yalcin. Identification of Mechanism of Action of DNA-Topoisomerase II Inhibitors by Molecular Modeling Studies, 20th European Symposium on Quantitative Structure-Activity Relationships (20th EuroQSAR), St-Petersburg, Russia, OC12: p52, 31 August - 4 September 2014. (Ağustos 2014)
  • smail Yalcin, Tugba Ertan Bolelli, Yaman Musdal, Kayhan Bolelli, Serap Yilmaz, Yasemin Aksoy, Bengt Mannervik, Ilkay Yildiz, Esin Aki Yalcin. Description of the Binding Site and GSH Conjugation Features of the New Human GST P1-1 Inhibitors, 20th European Symposium on Quantitative Structure-Activity Relationships (20th EuroQSAR), St-Petersburg, Russia, P150: p224, 31 August - 4 September 2014. (Ağustos 2014)
  • Ilkay Yildiz, Tugba Ertan-Bolelli, Serap Yilmaz, Sanaz Ataei, Kayhan Bolelli, Ozum Ozturk, Esin Karatas, Esin Aki-Yalcin, Ismail Yalcin. Molecular Modeling Studies on Some Benzazole Derivatives as Topoisomerase I Poison, 20th European Symposium on Quantitative Structure-Activity Relationships (20th EuroQSAR), St-Petersburg, Russia, P147: p221, 31 August - 4 September 2014. (Ağustos 2014)
  • Serap Yilmaz, Tugba Ertan Bolelli, Kayhan Bolelli, Ozum Ozturk, Sanaz Ataei, Ilkay Yildiz, Esin Aki Yalcin, Ismail Yalcin. Molecular Docking Studies of AcrB Trimeric Multidrug Efflux Pumps, 20th European Symposium on Quantitative Structure-Activity Relationships (20th EuroQSAR), St-Petersburg, Russia, P096: p170, 31 August - 4 September 2014. (Ağustos 2014)
  • Ilkay Yildiz, Sanaz Ataei, Serap Yilmaz, Tugba Ertan-Bolelli, Egemen Foto, Esin Aki-Yalcin, Ismail Yalcin. Molecular Modeling Studies On Some Topoisomerase I Inhibitors, 2nd International BAU-Drug Design Symposium 2014, Bahçeşehir University, Faculty of Medicine, Istanbul, Turkey, OP-1: p38-39, 17-19 April 2014. (Nisan 2014)
  • Esin Aki-Yalcin, Tugba Ertan-Bolelli, Tugba Taskin-Tok, Serap Yilmaz, Kayhan Bolelli, Ozum Ozturk, Ilkay Yildiz and Ismail Yalcin. Molecular Modeling Studies on DNA-Topoisomerase II Inhibitors, 2nd International BAU-Drug Design Symposium 2014, Bahçeşehir University, Faculty of Medicine, Istanbul, Turkey, IL-8: p18, 17-19 April 2014. (Nisan 2014)
  • Ismail Yalcin, Tugba Ertan-Bolelli, Yaman Musdal, Kayhan Bolelli, Serap Yilmaz, Yasemin Aksoy, Bengt Mannervik, Ilkay Yildiz, Esin Aki-Yalcin. Description of the Binding Site Features of Some Fused Heterocycles as New Human GST P1-1 Inhibitors, 2nd International BAU-Drug Design Symposium 2014, Bahçeşehir University, Faculty of Medicine, Istanbul, Turkey, CL-5: p9, 17-19 April 2014. (Nisan 2014)
  • Egemen Foto, Cigdem Ozen, Fatma Zilifdar, Serap Yilmaz, Sabiha Alper-Hayta, Ilkay Yildiz, Esin Aki-Sener, Ismail Yalcin, Nuran Diril. Inhibitory Effects of Some Benzoxazine Derivatives on Human DNA Topoisomerase I, 2nd International BAU-Drug Design Symposium 2014, Bahçeşehir University, Faculty of Medicine, Istanbul, Turkey, P-74: p155-156, 17-19 April 2014. (Nisan 2014)
  • Ismail Yalcin, Kayhan Bolelli, Serap Yilmaz, Tugba Ertan-Bolelli, Ozum Ozturk, Sanaz Ataei, Ilkay Yildiz, Esin Aki-Yalcin. CADD Studies on Chemotherapeutical Active Fused Heterocyclic Compounds, 9th AFMC International Medicinal Chemistry Symposium (AIMECS 13), The Grand Hotel, Taipei, Taiwan, S18-01: p55, 15-18 October 2013. (Ekim 2013)
  • Esin Aki-Yalcin, Tugba Ertan-Bolelli, Kayhan Bolelli, Serap Yilmaz, Ozum Ozturk, Tugba Taskin-Tok, Ilkay Yildiz and Ismail Yalcin. Rational Design of DNA-Topoisomerase Inhibitory Active Benzazoles as Antitumoral Agents, 9th AFMC International Medicinal Chemistry Symposium (AIMECS 13), The Grand Hotel, Taipei, Taiwan, O-37: p54, 15-18 October 2013. (Ekim 2013)
  • Esin Aki-Yalcin, Ismail Yalcin, Ilkay Yildiz, Tuğba Ertan-Bolelli, Kayhan Bolelli, Serap Yilmaz, Özüm Öztürk. Chemometrics in Drug Design, 2nd International Conference on New Trends in Chemometrics and Applications (NTCA-2013), Ankara University, Faculty of Pharmacy, Ankara, Turkey, IL-05: p7, 25-28 October 2013. (Ekim 2013)
  • Tugba Ertan-Bolelli, Ilkay Yildiz, Kayhan Bolelli, Serap Yilmaz, Sanaz Ataei, Ozum Ozturk, Selda Ozgen, Esin Aki, Ismail Yalcin. Molecular Docking Studies on Dihydropteroate Synthase Enzyme, Seventh International Symposium on Computational Methods in Toxicology and Pharmacology Integrating Internet Resources (CMTPI-2013), Seoul, South Korea, PO-C-09: p72, 8-12 October 2013. (Ekim 2013)
  • Kayhan Bolelli, Tuğba Ertan-Bolelli, Yaman Musdal, Serap Yilmaz, Ozum Ozturk, Yasemin Aksoy, Ilkay Yildiz, Esin Aki, Ismail Yalcin. Docking Studies on Glutathione S-Transferase P1-1 Enzyme, Seventh International Symposium on Computational Methods in Toxicology and Pharmacology Integrating Internet Resources (CMTPI-2013), Seoul, South Korea, PO-C-03: p66, 8-12 October 2013. (Ekim 2013)
  • Tugba Ertan-Bolelli, Ilkay Yildiz, Selda Ozgen, Kayhan Bolelli, Serap Yilmaz, Sanaz Ataei, Ozum Ozturk, Esin Aki-Yalcin, and Ismail Yalcin. Molecular Docking Studies on Enoyl-ACP Reductase Enzyme, 9th AFMC International Medicinal Chemistry Symposium (AIMECS 13), The Grand Hotel, Taipei, Taiwan, P1-05: p64, 15-18 October 2013. (Ekim 2013)
  • Serap Yilmaz, Ismail Yalcin, Tugba Ertan-Bolelli, Kayhan Bolelli, Ozum Ozturk, Sanaz Ataei, Ilkay Yildiz, and Esin Aki-Yalcin. Molecular Docking Studies on AcrB Trimeric Multidrug Efflux Pumps of Escherichia coli, 9th AFMC International Medicinal Chemistry Symposium (AIMECS 13), The Grand Hotel, Taipei, Taiwan, P1-04: p63, 15-18 October 2013. (Ekim 2013)
  • Kayhan Bolelli, Ismail Yalcin, Tugba Ertan-Bolelli, Serap Yilmaz, Ozum Ozturk, Yaman Musdal, Ilkay Yildiz and Esin Aki-Yalcin. Molecular Docking Studies of Glutathion S-Transferase Inhibitors, 9th AFMC International Medicinal Chemistry Symposium (AIMECS 13), The Grand Hotel, Taipei, Taiwan, P1-03: p62, 15-18 October 2013. (Ekim 2013)
  • J.B. Bhagyasree, Hema Tresa Varghese, C. Yohannan Panicker, Jadu Samuel, Christian Van Alsenoy, Serap Yilmaz, Ilkay Yildiz, Esin Aki. Quantum Mechanical and Spectroscopic (FT-IR, FT-Raman, 1H NMR And UV) Investigations of 2-(p-Nitrobenzyl) Benzoxazole, 2nd International Conference on New Trends in Chemometrics and Applications (NTCA-2013), Ankara University, Faculty of Pharmacy, Ankara, Turkey, PP-27: p55, October 25-28, 2013. (Ekim 2013)
  • Ozum OZTURK, Esin AKI-YALCIN, Tugba ERTAN-BOLELLI, Kayhan BOLELLI, Serap YILMAZ, Sanaz ATAEI, Ilkay YILDIZ, Ismail YALCIN. Common Feature Pharmacophore Generation of DNA Topoisomerase II Enzyme Inhibitors, 49th International Conference on Medicinal Chemistry (RICT-49), The Conference Center Nice Acropolis, Nice, France, HT094: p268, 3-5 July 2013. (Temmuz 2013)
  • Sanaz ATAEI, Serap YILMAZ, Ilkay YILDIZ, Tugba ERTAN-BOLELLI, Kayhan BOLELLI, Ozum OZTURK, Esin AKI-YALCIN, Ismail YALCIN. Molecular nDocking Studies of Some Benzazole Derivatives as DNA Topoisomerase I Inhibitors, 49th International Conference on Medicinal Chemistry (RICT-49), The Conference Center Nice Acropolis, Nice, France, HT006: p182, 3-5 July 2013. (Temmuz 2013)
  • Ismail Yalcin, Serap Yilmaz, Kayhan Bolelli, Tugba Ertan-Bolelli, Ilkay Yildiz, Esin Aki-Yalcin. Common Feature Pharmacophore Generation of Heterocyclic Compounds as Bacterial RND Efflux Pump Inhibitors, 1st International BAU-Drug Design Symposium 2013, Bahçeşehir University, Faculty of Medicine, Istanbul, Turkey, Lecture-2: p27, 21-23 March 2013. (Mart 2013)
  • Esin Aki, Tugba Taskin, Serap Yilmaz, Tugba Ertan-Bolelli, Kayhan Bolelli, Ozum Ozturk, Ilkay Yildiz, Ismail Yalcin, Yaman Musdal, Yasemin Aksoy. Molecular Modelling Studies on the Design of Chemotherapeutically Active Heterocyclic Compounds, 1st International BAU-Drug Design Symposium 2013, Bahçeşehir University, Faculty of Medicine, Istanbul, Turkey, Lecture-1: p26, 21-23 March 2013. (Mart 2013)
  • Kayhan BOLELLI, Ismail YALCIN, Tugba ERTAN-BOLELLI, Serap YILMAZ, Ozum OZTURK, Ilkay YILDIZ, Esin AKI-YALCIN. Docking Studies of Glutathion S-Transferase (GST) Inhibitors, 1st International BAU-Drug Design Symposium 2013, Bahçeşehir University, Faculty of Medicine, Istanbul, Turkey, P13: p65, 21-23 March 2013. (Mart 2013)
  • Ozum OZTURK, Esin AKI-YALÇIN, Tuğba ERTAN-BOLELLİ, Kayhan BOLELLİ, Serap YILMAZ, İlkay YILDIZ, İsmail YALÇIN. Docking Studies of Human Topoisomerase II Enzyme Inhibitors, 1st International BAU-Drug Design Symposium 2013, Bahçeşehir University, Faculty of Medicine, Istanbul, Turkey, P12: p64, 21-23 March 2013 (Mart 2013)
  • Serap YILMAZ, Ismail YALCIN, Tugba ERTAN-BOLELLI, Kayhan BOLELLI, Ozum OZTURK, Ilkay YILDIZ, Esin AKI-YALCIN. Molecular Modeling and Docking Studies of AcrB Trimeric Multidrug Efflux Pumps, 1st International BAU-Drug Design Symposium 2013, Bahçeşehir University, Faculty of Medicine, Istanbul, Turkey, P11: p63, 21-23 March 2013. (Mart 2013)
  • Esin Aki, Tugba Taskin, Ismail Yalcin, Yaman Musdal, Yasemin Aksoy, Serap Yilmaz, Tugba Ertan-Bolelli, Kayhan Bolelli, Ilkay Yildiz. Computational Drug Design Studies of Some New GST Inhibitory Active 2-Substituted Benzoxazoles and Benzothiazoles, EuroQSAR Knowledge Enabled Ligand Design, 19th European Symposium on Quantitative Structure-Activity Relationships (19th EuroQSAR), Vienna, Austria, P093: p156, 26-30 August 2012. (Ağustos 2012)
  • Serap Yilmaz, Sanaz Ataei, Ilkay Yildiz, Esin Aki, Ismail Yalcin. Pharmacophore Modelling of Some Fused Heterocyclic Compounds as HIV-1 Reverse Transcriptase Inhibitors, EuroQSAR Knowledge Enabled Ligand Design, 19th European Symposium on Quantitative Structure-Activity Relationships (19th EuroQSAR), Vienna, Austria, P083: p146, 26-30 August 2012. (Ağustos 2012)
  • Kayhan Bolelli, Serap Yilmaz, Ilkay Yildiz, Esin Aki, Ismail Yalcin. Common Feature Pharmacophore Generation of Bacterial AdeABC Efflux Pump Inhibitors, EuroQSAR Knowledge Enabled Ligand Design, 19th European Symposium on Quantitative Structure-Activity Relationships (19th EuroQSAR), Vienna, Austria, P078: p141, 26-30 August 2012. (Ağustos 2012)
  • Esin Akı, İsmail Yalçın, Ilkay Yildiz, Tuğba Taşkın, Tuğba Ertan-Bolelli, Serap Yilmaz, Kayhan Bolelli. Structure Based Drug Design Methods, 2nd International Conference on Computation for Science and Technology (ICCST-II), Nigde, Turkey, Invited Lec-7: p52, 09-11 July 2012. (Temmuz 2012)
  • Ismail Yalcin, Esin Aki, Ilkay Yildiz, Tugba Ertan-Bolelli, Kayhan Bolelli, and Serap Yilmaz. Computational Methods in Rational Drug Design, 2nd International Conference on Computation for Science and Technology (ICCST-II), Nigde, Turkey, Plenary Lec-5: p43, 09-11 July 2012. (Temmuz 2012)
  • Ismail Yalcin, Esin Aki, Ilkay Yildiz, Tugba Ertan-Bolelli, Kayhan Bolelli, and Serap Yilmaz. QSAR and Molecular Modeling Studies on Chemotherapeutic Active Benzazoles, 8th AFMC International Medicinal Chemistry Symposium (AIMECS 11), Keio Plaza Hotel, Tokyo, Japan, IL-B1: p8, 29 November-2 December 2011. (Kasım 2011)
  • Esin Aki, Ismail Yalcin, Ilkay Yildiz, Betul Tekiner-Gulbas, Tugba Ertan-Bolelli, Kayhan Bolelli, Serap Yilmaz, Sanaz Ataei, Özüm Öztürk. Chemometrics in Drug Design, 1st International Conference on New Trends in Chemometrics and Applications (NTCA-2011), Side, Antalya, Turkey, IL-05: p7, October 08-11, 2011. (Ekim 2011)
  • Serap Yılmaz, İlkay Yıldız, Esin Akı, İsmail Yalçın. 3D Pharmacophore Modelling of Some Fused Heterocyclic compounds as Topoisomerase II Inhibitor, 1st International Conference on New Trends in Chemometrics and Applications (NTCA-2011), Antalya PP-38: p65, 08-11 October 2011. (Ekim 2011)
  • Kayhan Bolelli, Serap Yılmaz, İsmail Yalçın, İlkay Yıldız, Esin Akı. QSAR Analysis of Some 2-Substituted Benzothiazoles as Antibacterial Agents against Multidrug-Resistant Staphylococcus aureus, 1st International Conference on New Trends in Chemometrics and Applications (NTCA-2011), Side, Antalya, Turkey, PP-37: p64, 08-11 October 2011. (Ekim 2011)
  • İlkay Yıldız, Serap Yılmaz, Sanaz Ataei, Esin Akı, İsmail Yalçın. Pharmacophore Analysis of Some Aromathecins as Topoisomerase I Inhibitor, 1st International Conference on New Trends in Chemometrics and Applications (NTCA-2011), Antalya, Turkey, PP-36: p63, 08-11 October 2011. (Ekim 2011)
  • Ismail Yalcin, Kayhan Bolelli, Serap Yilmaz, İlkay Yildiz, and Esin Aki-Yalcin. Common Feature Pharmacophore Generation of Heterocyclic Compounds against Efflux Pump Over-expressor Bacteria, 6th International Symposium on Computational Methods in Toxicology and Pharmacology Integrating Internet Resources (CMTPI-2011), Maribor, Slovenia, OC-21: p67, 03-07 September 2011. (Eylül 2011)
  • Esin Aki, Tugba Taskin, Yaman Musdal, Yasemin Aksoy, Serap Yilmaz, Tugba Ertan-Bolelli, Kayhan Bolelli, İlkay Yildiz, İsmail Yalcin. Docking Studies of GST Inhibitory Active 2-Substituted Benzazoles, 6th International Symposium on Computational Methods in Toxicology and Pharmacology Integrating Internet Resources (CMTPI-2011), Maribor, Slovenia, MT-07: p43, 03-07 September 2011. (Eylül 2011)
  • Esin Aki, İsmail Yalçin, İlkay Yildiz, Tugba Ertan-Bolelli, Kayhan Bolelli, Serap Yilmaz. Computational Drug Design Studies on Antitumoral Active Heterocyclic Compounds, 18th European Symposium on Quantitative Structure-Activity Relationships (18th EuroQSAR), Rhodes, Greece, OP27: p84, 19-24 September 2010. (Eylül 2010)
  • İlkay Yıldız, Sanaz Ataei, Serap Yılmaz, Egemen Foto, Tugba Ertan-Bolelli, Kayhan Bolelli, Nuran Diril, Esin Akı-Yalcin, İsmail Yalcin. Three-Dimensional Common-Feature Hypotheses on Benzoxazine Derivatives as Topoisomerase I Inhibitors, The 18th International Conference on Organic Synthesis (ICOS-18), Bergen, Norway, 377: p54, 1-6 August 2010. (Ağustos 2010)
  • Esin Akı, İsmail Yalçın, İlkay Yildiz, Tuğba Ertan-Bolelli, Kayhan Bolelli, Serap Yılmaz. Computer Aided Drug Design Studies on Chemotherapeutically Active Heterocyclic Compounds, Third International Meeting on Pharmacy & Pharmaceutical Sciences (IMPPS-3), Istanbul, Turkey, PL-2: p16, 9-12 June 2010. (Temmuz 2010)
  • Tugba Ertan-Bolelli, İlkay Yildiz, Kayhan Bolelli, Betül Tekiner-Gulbas, Serap Yilmaz, Özlem Temiz-Arpaci, Esin Aki and Ismail Yalcin. Pharmacophore Analysis on Some Benzoxazoles against Drug-Resistant Escherichia coli, Fifth International Symposium on Computational Methods in Toxicology and Pharmacology Integrating Internet Resources (CMTPI-2009), Istanbul, Turkey, PO-41: p108, 4-8 July 2009. (Temmuz 2009)

Ulusal Bilimsel Toplantılarda Sunulan ve Bildiri Kitabında Basılan Bildiriler

  • Egemen Foto, Fatma Zilifdar, Serap Yılmaz, İsmail Yalçın, Nuran Diril. Bir Seri 1,4-Benzoksazin-3-on Türevi Bileşiğin İn Vitro Anti-Kanser Etkileri ve Farmakofor Modellemesi, 23. Ulusal Biyoloji Kongresi, Gaziantep Üniversitesi, Gaziantep, Türkiye, 5-7 Eylül 2016. (Eylül 2016)
  • Tugba Taskin-Tok, Esin Akı, Ismail Yalcin, Ilkay Yildiz, Tugba Ertan-Bolelli, Kayhan Bolelli, Serap Yılmaz. Docking Studies of Topoisomerase II Inhibitors, Uluslararası Katılımlı 25. Ulusal Kimya Kongresi (UKK-25), Atatürk Üniversitesi, Erzurum, Türkiye, MS-013: p180, 27 Haziran - 02 Temmuz 2011. (Haziran 2011)
  • Esin Akı, İsmail Yalçın, İlkay Yıldız, Tugba Ertan-Bolelli, Kayhan Bolelli, Tugba Taşkın, Serap Yılmaz. Kemoterapötik Etkili Heterosiklik Bileşiklerin Bilgisayar Destekli İlaçTasarım Çalışmaları, Uluslararası Katılımlı 25. Ulusal Kimya Kongresi (UKK-25), Atatürk Üniversitesi, Erzurum, Türkiye, IL-009: p43, 27 Haziran - 02 Temmuz 2011. (Haziran 2011)

» Projeler

Ulusal » Diğer » Diğer (Ankara Üniversitesi Bilimsel Araştırma Projeleri)

Bazı Yeni Antitümör Etkili Heterosiklik Bileşiklerin Sentezi ve Moleküler Modellemesi
Proje Türü : Akademik     Görev : Araştırmacı     Kurum : Ankara Universitesi

Ulusal » Diğer » Diğer (Ankara Üniversitesi Bilimsel Araştırma Projeleri)

Bazı Yeni DNA Topoizomeraz Etkili İnhibitör Benzotiyazol Türevlerinin Sentezi
Proje Türü : Altyapı     Görev : Araştırmacı     Kurum : Ankara Üniversitesi

» Verdiği Dersler

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İlaç Etken Madde Tasarımı

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